SCHEMBL9846127

SCHEMBL9846127

COc1cc([N+](=O)[O-])c(=O)[nH]c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
CYP3A4 P08684 2/20 0.47
ALOX15 P16050 1/20 0.47
PRKDC P78527 1/20 0.47
HSD17B10 Q99714 1/20 0.47
GAA P10253 1/20 0.45
PDE3B Q13370 6/20 0.45
PDE3A Q14432 6/20 0.45
TDP1 Q9NUW8 3/20 0.44
GRIN2D O15399 3/20 0.43
GRIN3B O60391 3/20 0.43
GRIN1 Q05586 3/20 0.43
GRIN2A Q12879 3/20 0.43
GRIN2B Q13224 3/20 0.43
GRIN2C Q14957 3/20 0.43
GRIN3A Q8TCU5 3/20 0.43
BLM P54132 2/20 0.43
LMNA P02545 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL215905 0.78 KDM4E (0.52) MAPTKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL28457504 0.75 KDM4E (0.49) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL210330 0.75 ALDH1A1 (0.68) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL10778338 0.75 ALDH1A1 (0.62) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL29800558 0.75 ALDH1A1 (0.68) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL9332963 0.74 KDM4E (0.47) MAPTKDM4ECYP3A4GAAGRIN2D
SCHEMBL9432382 0.72 KDM4E (0.46) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL27944806 0.72 GRIN2D (0.67) MAPTCYP3A4ALOX15TDP1GRIN2D
SCHEMBL3294994 0.72 ALDH1A1 (0.59) MAPTKDM4EALDH1A1CYP3A4ALOX15
SCHEMBL11251378 0.72 ALDH1A1 (0.55) MAPTKDM4EALDH1A1CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed
US-4131677-A Anti-inflammatory oxazolo [5,4-b]pyridines MERCK & CO., INC. (US) 1978-12-26 US disclosed
US-4038396-A ANTIPYRETICS, ANALGESICS MERCK & CO., INC. (US) 1977-07-26 US disclosed