SCHEMBL9848571

SCHEMBL9848571

Nc1nnc(-c2cc(Cl)c([N+](=O)[O-])c(Cl)c2Cl)c(N)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.48
SCN2A Q99250 2/20 0.48
CYP2D6 P10635 1/20 0.48
MAOA P21397 1/20 0.48
MAPK1 P28482 1/20 0.48
ADRA1A P35348 1/20 0.48
SCN4A P35499 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
PDE3A Q14432 1/20 0.48
SCN5A Q14524 1/20 0.48
SCN3A Q9NY46 1/20 0.48
SCN10A Q9Y5Y9 1/20 0.48
DHFR P00374 1/20 0.40
ALDH1A1 P00352 3/20 0.38
TSHR P16473 2/20 0.38
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5070878 0.79 DHFR (0.56) SCN2ADHFRALDH1A1TSHRNPC1
SCHEMBL9848562 0.77 SCN9A (0.57) SCN9ASCN2ACYP2D6MAOAMAPK1
SCHEMBL5072690 0.76 NCOA1 (0.41) CYP2D6DHFRALDH1A1TSHRCCNA2
SCHEMBL978226 0.71 SCN9A (0.61) SCN9ASCN2ACYP2D6MAOAMAPK1
SCHEMBL30413401 0.71 SCN9A (0.61) SCN9ASCN2ACYP2D6MAOAMAPK1
SCHEMBL8903239 0.70 SCN9A (0.55) SCN9ASCN2ACYP2D6MAOAMAPK1
SCHEMBL7377151 0.69 SCN2A (0.47) SCN9ASCN2ASCN5ASCN3ASCN10A
SCHEMBL9848578 0.69 SCN9A (0.54) SCN9ASCN2ACYP2D6MAOAMAPK1
SCHEMBL6374569 0.69 SCN9A (0.58) SCN9ASCN2ACYP2D6MAOAMAPK1
SCHEMBL16854426 0.69 SCN9A (0.58) SCN9ASCN2ACYP2D6MAOAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0459829-A1 Pharmacologically active CNS compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed