SCHEMBL9849428

SCHEMBL9849428

Cc1c(CCC(C)n2ccnc2)c(N)nc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
TLR8 Q9NR97 6/20 0.41
TLR7 Q9NYK1 2/20 0.39
CYP17A1 P05093 4/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
HRH2 P25021 1/20 0.37
ADRA1D P25100 1/20 0.37
HTR2A P28223 1/20 0.37
ADORA2A P29274 1/20 0.37
ADRA1A P35348 1/20 0.37
NUDT1 P36639 1/20 0.37
HTR2B P41595 1/20 0.37
PDE4D Q08499 1/20 0.37
KCNH2 Q12809 1/20 0.37
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849506 0.79 KDM4E (0.39) KDM4ETLR7CYP17A1LMNAPOLB
SCHEMBL9849295 0.78 TSHR (0.55) TLR8CYP19A1
SCHEMBL9849636 0.77 TSHR (0.54) TLR8
SCHEMBL9849555 0.75 ALDH1A1 (0.43) TLR8TLR7LMNAPOLBHRH2
SCHEMBL5305103 0.73 KDM4E (0.55) KDM4ECYP17A1POLBCYP19A1
SCHEMBL16836321 0.70 TLR8 (0.74) TLR8TLR7
Dimethylamine SCHEMBL10651852 0.70 KDM4E (0.54) KDM4ECYP17A1POLBCYP19A1
SCHEMBL9849435 0.70 KDM4E (0.49) KDM4ELMNA
SCHEMBL11017730 0.66 KDM4E (0.50) KDM4ECYP17A1CYP19A1
SCHEMBL16836395 0.66 TLR8 (0.74) KDM4ETLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed