SCHEMBL9849541

SCHEMBL9849541

Nc1nc2cccc(CCCCn3ccnc3)c2c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.51
TBXAS1 P24557 1/20 0.51
POLB P06746 1/20 0.46
TSHR P16473 1/20 0.45
GAA P10253 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
SOD1 P00441 1/20 0.43
HMOX1 P09601 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849395 0.96 CYP19A1 (0.52) CYP19A1TBXAS1POLBTSHRGAA
SCHEMBL9849700 0.84 CYP19A1 (0.51) CYP19A1TBXAS1POLBTSHRGAA
SCHEMBL9849690 0.80 POLB (0.44) CYP19A1TBXAS1POLBTSHRALDH1A1
SCHEMBL9849636 0.78 TSHR (0.54) TSHRGAAALDH1A1GSK3AGSK3B
SCHEMBL11247886 0.76 POLB (0.68) CYP19A1TBXAS1POLBGAASOD1
SCHEMBL9849511 0.76 TLR8 (0.57) CYP19A1TBXAS1TSHRSOD1
SCHEMBL9849506 0.75 KDM4E (0.39) CYP19A1TBXAS1POLB
SCHEMBL9849295 0.74 TSHR (0.55) CYP19A1TSHRGAAALDH1A1GSK3A
SCHEMBL9849881 0.72 GAA (0.55) CYP19A1TBXAS1TSHRGAAALDH1A1
SCHEMBL9849597 0.71 SOD1 (0.48) CYP19A1POLBTSHRALDH1A1SOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed