SCHEMBL9851617

SCHEMBL9851617

Cc1ccc(S(=O)(=O)N2CC3(CCN(C)C3)C2)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.60
CYP1A2 P05177 2/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
PKM P14618 3/20 0.54
HTT P42858 2/20 0.53
ALDH1A1 P00352 1/20 0.53
POLB P06746 1/20 0.53
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.49
GAA P10253 2/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
LMNA P02545 1/20 0.48
NAMPT P43490 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16572126 0.87 PKM (0.56) TSHRCYP1A2CYP3A4CYP2D6PKM
SCHEMBL9851568 0.84 PKM (0.63) TSHRPKMHTTALDH1A1POLB
SCHEMBL20840919 0.83 PKM (0.59) TSHRCYP1A2PKMHTTALDH1A1
SCHEMBL18047962 0.81 PKM (0.66) TSHRPKMHTTALDH1A1POLB
SCHEMBL14149366 0.81 PKM (0.59) TSHRCYP1A2CYP3A4CYP2D6PKM
SCHEMBL21595328 0.79 PKM (0.54) TSHRCYP1A2CYP3A4CYP2D6PKM
SCHEMBL21060157 0.78 PKM (0.53) TSHRPKMHTTALDH1A1POLB
SCHEMBL196221 0.78 PKM (0.56) TSHRPKMHTTALDH1A1POLB
SCHEMBL825032 0.77 PKM (0.59) TSHRPKMHTTALDH1A1POLB
SCHEMBL5900909 0.77 PKM (0.51) TSHRCYP3A4PKMHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417631-A2 Condensed diazepinones, process for their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1991-03-20 EP disclosed