SCHEMBL9851624

SCHEMBL9851624

Cc1scc2c1N(C(=O)N1CCC3(CN(C)C3)C1)c1ccccc1NC2=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.62
CYP2C9 P11712 2/20 0.62
CYP2C19 P33261 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2D6 P10635 2/20 0.62
CYP3A4 P08684 1/20 0.62
TSHR P16473 1/20 0.62
L3MBTL1 Q9Y468 1/20 0.62
LMNA P02545 3/20 0.61
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CHRM1 P11229 5/20 0.35
CHRM2 P08172 4/20 0.35
CHRM4 P08173 4/20 0.35
CHRM3 P20309 4/20 0.35
USP2 O75604 1/20 0.35
CHRM5 P08912 1/20 0.35
GMNN O75496 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9851561 0.96 CYP3A4 (0.60) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851853 0.95 CYP3A4 (0.61) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851636 0.95 ALDH1A1 (0.63) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851650 0.92 ALDH1A1 (0.65) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851638 0.92 ALDH1A1 (0.63) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851639 0.91 ALDH1A1 (0.58) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851607 0.88 CYP3A4 (0.57) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851647 0.88 ALDH1A1 (0.60) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851579 0.87 ALDH1A1 (0.58) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9851620 0.85 CYP2D6 (0.56) ALDH1A1CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0417631-A2 Condensed diazepinones, process for their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1991-03-20 EP disclosed