SCHEMBL9851680

SCHEMBL9851680

COC(=O)N(C)CC#CCNCCCCCO

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PAOX Q6QHF9 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
CHRM1 P11229 1/20 0.33
POLB P06746 1/20 0.32
ACHE P22303 6/20 0.30
CYP4F2 P78329 1/20 0.30
CYP4A11 Q02928 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9851686 0.98 CHRM1 (0.34) PAOXTDP1CHRM1POLB
SCHEMBL9851792 0.80 CHRM1 (0.37) PAOXCHRM1ACHE
SCHEMBL9779511 0.79 CHRM1 (0.34) CHRM1
SCHEMBL9779592 0.78 CHRM1 (0.35) CHRM1
SCHEMBL9779487 0.74 CHRM1 (0.59) CHRM1
SCHEMBL9779728 0.69 CHRM1 (0.44) CHRM1
SCHEMBL11728208 0.69 CHRM1 (0.53) PAOXCHRM1
SCHEMBL22282294 0.68 LMNA (0.40) CHRM1POLBCYP4F2CYP4A11
SCHEMBL20373148 0.68 LMNA (0.35) TDP1
SCHEMBL9779570 0.67 CHRM1 (0.37) CHRM1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0411616-A1 4-(N-substituted amino)-2-butynyl-1-carbamates and thiocarbamates and derivatives thereof as centrally acting muscarinic agents WARNER-LAMBERT COMPANY (US) 1991-02-06 EP disclosed