SCHEMBL9851994

SCHEMBL9851994

CC[15N]1CCC(=NO)c2ccn(CCCCN3CCC(C(=O)c4ccc(F)cc4)CC3)c2C1=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
DRD2 P14416 1/20 0.46
HTR7 P34969 2/20 0.45
HTR2C P28335 3/20 0.44
HTR6 P50406 1/20 0.44
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9041369 1.00 HTR2A (0.46) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9039895 0.94 HTR2A (0.47) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9040040 0.94 HTR2A (0.46) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL6993587 0.92 HTR2A (0.47) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL6993584 0.92 HTR2A (0.47) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9041322 0.91 DRD2 (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9041080 0.90 DRD2 (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9039482 0.90 HTR2A (0.49) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9039019 0.89 DRD2 (0.53) HTR2AKDM4ECYP1A2CYP3A4CYP2D6
SCHEMBL9039858 0.89 HTR2A (0.54) HTR2AKDM4ECYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0441349-A1 Pyrroloazepine derivatives SUNTORY LIMITED (JP) 1991-08-14 EP disclosed