SCHEMBL9853589

SCHEMBL9853589

Nc1ccnc(-c2ccc3ccccc3c2)c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.49
HTR5A P47898 1/20 0.49
ADORA2A P29274 3/20 0.47
ADORA1 P30542 3/20 0.47
CYP1A2 P05177 1/20 0.46
SRC P12931 5/20 0.46
ABL1 P00519 4/20 0.46
MAPK9 P45984 2/20 0.45
MAPK10 P53779 2/20 0.45
DHFR P00374 1/20 0.45
MAPK8 P45983 1/20 0.45
KDM4E B2RXH2 2/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
AR P10275 1/20 0.44
MAPT P10636 1/20 0.44
NFKB1 P19838 1/20 0.44
RAB9A P51151 1/20 0.44
GFER P55789 1/20 0.44
NFKB2 Q00653 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9853594 0.87 CCNC (0.46) HTR2BHTR5AADORA2AADORA1SRC
Maleic Acid SCHEMBL9853592 0.87 CCNC (0.46) HTR2BHTR5AADORA2AADORA1SRC
SCHEMBL29419535 0.79 ADORA2A (0.51) HTR2BHTR5AADORA2AADORA1CYP1A2
SCHEMBL27843373 0.78 CDK5 (0.45) HTR2BHTR5AADORA2AADORA1MAPK9
SCHEMBL4058635 0.77 CDK5 (0.47) HTR2BHTR5AADORA2AADORA1CYP1A2
SCHEMBL31695983 0.77 MAPKAPK2 (0.45) HTR2BHTR5AADORA2AADORA1CYP1A2
SCHEMBL19432619 0.77 ALK (0.45) HTR2BHTR5AADORA2AADORA1SRC
SCHEMBL729774 0.75 HTR2B (0.59) HTR2BHTR5AADORA2AADORA1CYP1A2
SCHEMBL29445836 0.75 HTR2B (0.59) HTR2BHTR5AADORA2AADORA1CYP1A2
SCHEMBL18703800 0.73 DYRK1A (0.57) CYP1A2SRCABL1MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0405426-A2 Naphthylamino- and naphthyloxy-pyridinamines and related compounds, a process for their preparation and their use as dermatological agents HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-01-02 EP disclosed