SCHEMBL9856784

SCHEMBL9856784

CC(C)c1nc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)n1CCC(O)CC(O)CC(=O)O.[NaH]

nearest known ligand 0.80

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 12/20 0.63
NR1I2 O75469 1/20 0.54
ABCB11 O95342 1/20 0.54
RHOC P08134 1/20 0.54
CYP3A4 P08684 1/20 0.54
THRB P10828 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC2 Q92769 1/20 0.54
NR1H4 Q96RI1 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
ABCG2 Q9UNQ0 1/20 0.54
SLCO1B1 Q9Y6L6 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857125 0.99 HMGCR (0.64) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9856946 0.96 HMGCR (0.61) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9856838 0.95 HMGCR (0.60) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9857159 0.94 HMGCR (0.59) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9857215 0.94 HMGCR (0.59) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9856789 0.89
SCHEMBL9856756 0.84 HMGCR (0.52) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL4103858 0.84 HMGCR (0.51) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9856801 0.83 HMGCR (0.65) HMGCR
SCHEMBL4098730 0.83 HMGCR (0.51) HMGCRNR1I2ABCB11RHOCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0436851-A1 Compounds active as inhibitors of the enzyme HMG-CoA reductase and pharmaceutical compositions containing them ZAMBON GROUP S.p.A. (IT) 1991-07-17 EP disclosed