SCHEMBL9856840

SCHEMBL9856840

Cc1nc(-c2ccccc2)n(CCC(O)CC(O)CC(=O)O)c1C

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 11/20 0.54
NR1I2 O75469 1/20 0.44
ABCB11 O95342 1/20 0.44
RHOC P08134 1/20 0.44
CYP3A4 P08684 1/20 0.44
THRB P10828 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
NR1H4 Q96RI1 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
SLCO1B1 Q9Y6L6 1/20 0.44
MMP2 P08253 1/20 0.40
MMP9 P14780 1/20 0.40
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
MMP14 P50281 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9482214 0.82 KDM4E (0.59) HMGCR
SCHEMBL9857442 0.80 FAAH (0.54) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL9856979 0.79 HMGCR (0.45) HMGCRABCB11
SCHEMBL9856973 0.79 HMGCR (0.45) HMGCRABCB11
SCHEMBL4977553 0.78 HMGCR (0.48) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL5518690 0.78 HMGCR (0.47) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL5994174 0.77 HMGCR (0.64) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL5225591 0.77 HMGCR (0.64) HMGCRNR1I2ABCB11RHOCCYP3A4
SCHEMBL5224981 0.76 HMGCR (0.84) HMGCR
SCHEMBL5224248 0.76 HMGCR (0.88) HMGCRNR1I2ABCB11RHOCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0436851-A1 Compounds active as inhibitors of the enzyme HMG-CoA reductase and pharmaceutical compositions containing them ZAMBON GROUP S.p.A. (IT) 1991-07-17 EP disclosed