SCHEMBL9859142

SCHEMBL9859142

Cc1ccc(N=C=S)cc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY6 Q15077 2/20 0.41
CYP3A4 P08684 3/20 0.40
MIF P14174 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
TRPA1 O75762 1/20 0.40
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
PNMT P11086 1/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
USP2 O75604 3/20 0.37
MAPT P10636 3/20 0.37
HPGD P15428 3/20 0.37
HSD17B10 Q99714 3/20 0.37
LTA P01374 2/20 0.37
P2RX3 P56373 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30016097 1.00 P2RY6 (0.41) P2RY6CYP3A4MIFCA1CA2
SCHEMBL2886976 0.84 P2RY6 (0.41) P2RY6CYP3A4MIFCA1CA2
SCHEMBL3036837 0.81 P2RY6 (0.45) P2RY6CYP3A4MIFCA1CA2
SCHEMBL6154714 0.81 P2RY6 (0.45) P2RY6CYP3A4MIFCA1CA2
SCHEMBL419490 0.80 CYP3A4 (0.63) CYP3A4TRPA1MEN1KMT2ANPC1
SCHEMBL484205 0.78 CYP3A4 (0.60) P2RY6CYP3A4MIFCA1CA2
SCHEMBL29463953 0.78 CYP3A4 (0.60) P2RY6CYP3A4MIFCA1CA2
SCHEMBL13559510 0.76 P2RY6 (0.41) P2RY6CYP3A4MIFCA1CA2
SCHEMBL13210766 0.76 TDP1 (0.42) P2RY6CYP3A4MIFCA1CA2
SCHEMBL15221651 0.76 P2RY6 (0.41) P2RY6CYP3A4MIFCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153127-B1 N-ARYL-3-ARYL-4,5-DIHYDRO-1H-PYRAZOLE-1-CARBOXAMIDES, PROCESSES FOR THEIR PRODUCTION, INSECTICIDAL COMPOSITIONS CONTAINING THEM AND METHODS FOR COMBATTING INSECTS ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
US-4863947-A PESTICIDES, INSECTICIDES ROHM AND HAAS (US) 1989-09-05 US disclosed
US-4663341-A Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides ROHM AND HAAS COMPANY (US) 1987-05-05 US disclosed
EP-0153127-A2 N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamides, processes for their production, insecticidal compositions containing them and methods for combatting insects ROHM AND HAAS COMPANY (US) 1985-08-28 EP disclosed