SCHEMBL9859233

SCHEMBL9859233

O=C=Nc1ccc(C(F)(F)F)c(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
NOTUM Q6P988 1/20 0.41
CYP3A4 P08684 2/20 0.41
TRPA1 O75762 1/20 0.41
TSHR P16473 1/20 0.37
CYP1A2 P05177 1/20 0.32
KIF11 P52732 1/20 0.30
HTR3E A5X5Y0 1/20 0.30
HTR3B O95264 1/20 0.30
HTR3A P46098 1/20 0.30
HTR3D Q70Z44 1/20 0.30
HTR3C Q8WXA8 1/20 0.30
CES2 O00748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL281622 0.86 MAPK1 (0.43) MAPK1TDP1NOTUMCYP3A4TRPA1
SCHEMBL11878079 0.85 MAPK1 (0.46) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL1555041 0.83 MAPK1 (0.47) MAPK1TDP1NOTUMCYP3A4TRPA1
SCHEMBL1493109 0.80 CYP3A4 (0.55) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL30196175 0.80 KIF11 (0.45) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL4462791 0.80 KIF11 (0.45) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL856525 0.79 MAPK1 (0.61) MAPK1TDP1NOTUMCYP3A4TRPA1
SCHEMBL7177146 0.78 MAPK1 (0.46) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL11517806 0.77 MAPK1 (0.52) MAPK1TDP1CYP3A4TRPA1TSHR
SCHEMBL3104369 0.76 CYP3A4 (0.50) MAPK1TDP1CYP3A4TRPA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153127-B1 N-ARYL-3-ARYL-4,5-DIHYDRO-1H-PYRAZOLE-1-CARBOXAMIDES, PROCESSES FOR THEIR PRODUCTION, INSECTICIDAL COMPOSITIONS CONTAINING THEM AND METHODS FOR COMBATTING INSECTS ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
US-4863947-A PESTICIDES, INSECTICIDES ROHM AND HAAS (US) 1989-09-05 US disclosed
US-4663341-A Insecticidal n-aryl-3-aryl-4,5-dihydro-1h-pyrazole-1-carboxamides ROHM AND HAAS COMPANY (US) 1987-05-05 US disclosed
EP-0153127-A2 N-aryl-3-aryl-4,5-dihydro-1H-pyrazole-1-carboxamides, processes for their production, insecticidal compositions containing them and methods for combatting insects ROHM AND HAAS COMPANY (US) 1985-08-28 EP disclosed