SCHEMBL9860009

SCHEMBL9860009

COc1cc2c(cc1/C(C)=C/c1ccc(OC(=O)O)cc1)C(C)(C)CCC2(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 16/20 0.56
RARB P10826 16/20 0.56
RARG P13631 15/20 0.56
RARA P10276 11/20 0.56
RXRB P28702 6/20 0.56
RXRG P48443 6/20 0.56
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
CYP26A1 O43174 1/20 0.49
GMNN O75496 1/20 0.49
USP2 O75604 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
NFKB1 P19838 1/20 0.49
CYP2C19 P33261 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11212795 0.87 RARB (0.74) RXRARARBRARGRARARXRB
SCHEMBL11221509 0.87 RARB (0.74) RXRARARBRARGRARARXRB
SCHEMBL8776401 0.85 RXRA (0.54) RXRARARBRARGRARARXRB
SCHEMBL7135063 0.85 RXRA (0.54) RXRARARBRARGRARARXRB
SCHEMBL9860395 0.84 RARB (0.52) RXRARARBRARGRARARXRB
SCHEMBL9860392 0.84 RARB (0.52) RXRARARBRARGRARARXRB
Methyl Alcohol SCHEMBL10474586 0.83 RARB (0.51) RXRARARBRARGRARARXRB
SCHEMBL7081825 0.80 RARB (0.57) RXRARARBRARGRARARXRB
SCHEMBL7081821 0.80 RARB (0.57) RXRARARBRARGRARARXRB
SCHEMBL10711895 0.77 RARB (0.48) RXRARARBRARGRARARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5055622-A For treating neoplasms and dermatoses HOFFMANN-LA ROCHE INC. (US) 1991-10-08 US disclosed
US-5030765-A Skin disorders, anititumor agents HOFFMANN-LA ROCHE INC. (US) 1991-07-09 US disclosed
US-5030764-A Antitumor agents; treatment of skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-07-09 US disclosed
US-5001276-A Novel tetrahydronaphthalene and indane derivatives HOFFMANN-LA ROCHE INC. (US) 1991-03-19 US disclosed
US-4990703-A Novel tetrahydronaphthalene and indane derivatives HOFFMANN-LA ROCHE INC. (US) 1991-02-05 US disclosed
US-4935560-A ANTITUMOR AGENTS; SKIN DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-06-19 US disclosed
US-4870219-A NEOPLASMS, DERMATOSES HOFFMANN-LA ROCHE INC. (US) 1989-09-26 US disclosed