SCHEMBL9860209

SCHEMBL9860209

CC(Cc1ccccc1)C(N)N

nearest known ligand 0.75

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.75
TAAR1 Q96RJ0 4/20 0.67
SLC6A2 P23975 2/20 0.67
SIGMAR1 Q99720 2/20 0.67
MAOA P21397 1/20 0.67
SLC6A4 P31645 1/20 0.67
SLC6A3 Q01959 1/20 0.67
CYP2A6 P11509 1/20 0.67
ADORA2A P29274 1/20 0.67
ADORA1 P30542 1/20 0.67
TRPA1 O75762 2/20 0.59
EPHX1 P07099 1/20 0.58
SLC18A2 Q05940 1/20 0.50
ANPEP P15144 1/20 0.50
ALPI P09923 1/20 0.48
PKM P14618 1/20 0.48
PTGS1 P23219 1/20 0.48
XIAP P98170 1/20 0.48
SLC7A5 Q01650 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23869573 0.86 CYP2D6 (1.00) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL15834911 0.86 CYP2D6 (1.00) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL30934 0.85 TRPA1 (0.77) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
Water SCHEMBL3896311 0.82 TRPA1 (0.74) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL1140503 0.82 TRPA1 (0.74) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL1396351 0.82 CYP2D6 (0.69) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL13243863 0.80 CYP2D6 (0.67) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL13243866 0.80 CYP2D6 (0.67) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL13243865 0.80 CYP2D6 (0.67) CYP2D6TAAR1SLC6A2SIGMAR1MAOA
SCHEMBL13243599 0.80 CYP2D6 (0.67) CYP2D6TAAR1SLC6A2SIGMAR1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3774716-B1 PROCESS FOR THE PREPARATION OF AMINES BASF SE (DE) 2022-03-16 EP disclosed
US-5021220-A Haluaromatic compound, water-soluble acid, copper salt acid-stable reducing agent MALLINCKRODT, INC. (US) 1991-06-04 US disclosed
US-4942231-A CATALYTIC HALOGENATION IN THE PRESENCE OF A REDUCING AGENT AND ACID MEDIUM MALLINCKRODT, INC. (US) 1990-07-17 US disclosed
EP-0165630-A2 Method of preparing a chlorinated, brominated, radiobrominated, iodinated and/or radioiodinated, aromatic or heteroaromatic compound, as well as a kit for preparing a diagnostic composition on the basis of this compound MALLINCKRODT, INC.(a Missouri corporation) (US) 1985-12-27 EP disclosed