SCHEMBL9861334

SCHEMBL9861334

Cc1cc(C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F)cc(C)c1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.47
ESR2 Q92731 2/20 0.47
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
PTGS1 P23219 5/20 0.34
PTGS2 P35354 5/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2B6 P20813 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPT P10636 3/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALOX5 P09917 3/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 2/20 0.32
AR P10275 1/20 0.31
XBP1 P17861 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL697863 0.98 ESR1 (0.48) ESR1ESR2CA1CA2PTGS1
SCHEMBL9861946 0.83 CYP2C9 (0.52) ESR1ESR2CA1CA2PTGS1
SCHEMBL22032589 0.83 ERN1 (0.42) ESR1ESR2CYP1A2CYP2C9CYP3A4
SCHEMBL10825969 0.79 LMNA (0.43) LMNA
SCHEMBL9861493 0.79 POLB (0.45) CYP3A4LMNAALDH1A1
SCHEMBL5958687 0.79 POLB (0.45) CYP3A4LMNAALDH1A1
SCHEMBL5958703 0.79 POLB (0.45) CYP3A4LMNAALDH1A1
SCHEMBL7157861 0.79 ESR1 (0.52) ESR1ESR2AR
SCHEMBL2837831 0.78 ESR1 (0.45) ESR1ESR2CA1CA2PTGS1
SCHEMBL9861307 0.77 SMN1; SMN2 (0.39) CA1CA2CYP1A2CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
EP-0336371-A2 Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-11 EP disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed
US-4845258-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-07-04 US disclosed
US-4804774-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804772-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-02-14 US disclosed
US-4804773-A Production of gem-disubstituted cyclohexadienones ETHYL CORPORATION (US) 1989-02-14 US disclosed