SCHEMBL9863186

SCHEMBL9863186

Cc1c(N=C=O)cc(N=C=O)cc1C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.49
TRPA1 O75762 1/20 0.49
TDP1 Q9NUW8 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15317 0.82 CYP3A4 (0.61) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL6057020 0.81 CYP3A4 (0.59) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL38512 0.79 CYP3A4 (0.41) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL163362 0.77 CYP3A4 (0.60) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL2585906 0.76 CYP3A4 (0.59) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL31425155 0.76 CYP3A4 (0.59) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL10526387 0.76 CA2 (0.50) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL1483790 0.75 CYP3A4 (0.41) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL14812425 0.74 CYP3A4 (0.52) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL8608054 0.74 CYP3A4 (0.52) CYP3A4TRPA1TDP1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0370408-A1 Process for the preparation of polyisocyanate prepolymers and polyurethanes and resulting compositions AIR PRODUCTS AND CHEMICALS, INC. (US) 1990-05-30 EP claimed
EP-0244778-B1 MONO-TERTIARY-ALKYLATED TOLUENEDIISO-CYANATES AND DERIVATIVES AIR PRODUCTS AND CHEMICALS, INC. (US) 1991-10-16 EP disclosed
EP-0370408-A1 Process for the preparation of polyisocyanate prepolymers and polyurethanes and resulting compositions AIR PRODUCTS AND CHEMICALS, INC. (US) 1990-05-30 EP disclosed
EP-0303914-A2 Urethane linked hydroxy aromatic amines AIR PRODUCTS AND CHEMICALS, INC. (US) 1989-02-22 EP disclosed
EP-0283868-A2 Process for producing polyurethane/urea elastomers AIR PRODUCTS AND CHEMICALS, INC. (US) 1988-09-28 EP disclosed
EP-0275030-A1 Urethane linked hydroxy aromatic isocyanates AIR PRODUCTS AND CHEMICALS, INC. (US) 1988-07-20 EP disclosed
US-4724256-A REACTING AROMATIC DIISOCYANATE AND ALIPHATIC POLYOL, CONTROLLING TEMPERATURE AND TIME TO PRODUCE ONE URETHANE LINKAGE AIR PRODUCTS AND CHEMICALS, INC. (US) 1988-02-09 US disclosed
US-4722989-A URETHANE-LINKED TOLUENEDIISOCYANATE, DIAMINE CHAIN EXTENSION AIR PRODUCTS AND CHEMICALS, INC. (US) 1988-02-02 US disclosed
EP-0244778-A1 Mono-tertiary-alkylated toluenediiso-cyanates and derivatives AIR PRODUCTS AND CHEMICALS, INC. (US) 1987-11-11 EP disclosed