SCHEMBL9866016

SCHEMBL9866016

CC12CCCC(CN1)N(c1cc3c(cc1F)c(=O)c(C(=O)O)cn3C1CC1)C2

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
ALDH1A1 P00352 4/20 0.57
LMNA P02545 3/20 0.56
HPGD P15428 2/20 0.56
HSD17B10 Q99714 2/20 0.56
TOP2B Q02880 2/20 0.56
CYP1A2 P05177 1/20 0.56
TOP2A P11388 1/20 0.56
CYP2C9 P11712 1/20 0.56
MAPT P10636 1/20 0.56
PIK3CG P48736 7/20 0.47
PIK3CD O00329 5/20 0.47
PIK3R1 P27986 5/20 0.47
PIK3CA P42336 5/20 0.47
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HRH3 Q9Y5N1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866559 0.84 TOP2A (0.50) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9864761 0.82 KDM4E (0.54) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9865688 0.82 ALDH1A1 (0.54) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9142889 0.80 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9142880 0.80 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9142884 0.80 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9866284 0.79 KDM4E (0.61) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9150397 0.78 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9150407 0.78 KDM4E (0.62) KDM4EALDH1A1LMNAHPGDHSD17B10
SCHEMBL9670775 0.78 KDM4E (0.64) KDM4EALDH1A1LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992546-A Process for preparing 6,8-diazabicyclo[3.2.2]nonane derivatives WARNER-LAMBERT COMPANY (US) 1991-02-12 US disclosed
US-4968799-A Antibacterial agents WARNER-LAMBERT COMPANY (US) 1990-11-06 US disclosed
US-4962108-A A QUIN-4-ONE HAVING THE FOLLOWING RING SUBSTITUENTS; 1-ALKYL OR PHENYL, 3-CARBOXY DERIVATIVE, 6-FLUORO AND 8-BRIDGED N-HETEROCYCLIC RING WARNER-LAMBERT COMPANY (US) 1990-10-09 US disclosed
US-4923879-A CARBOXYLIC ACID DERIVATIVES WITH BRIDGED SIDECHAINS WARNER-LAMBERT COMPANY (US) 1990-05-08 US disclosed
EP-0305744-A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-03-08 EP disclosed