SCHEMBL9866176

SCHEMBL9866176

CS(=O)(=O)Nc1ccc(OCC(O)CN2CCN(c3ncccn3)CC2)cc1

nearest known ligand 0.73

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.73
ADRB1 P08588 7/20 0.73
ADRB3 P13945 7/20 0.73
KCNH2 Q12809 1/20 0.70
KDM4E B2RXH2 2/20 0.59
MAPT P10636 3/20 0.52
NPSR1 Q6W5P4 1/20 0.52
HSP90AB1 P08238 1/20 0.52
PRMT5 O14744 1/20 0.51
WDR77 Q9BQA1 1/20 0.51
GLA P06280 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
USP2 O75604 1/20 0.50
TSHR P16473 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2019520 0.89 ADRB2 (0.72) ADRB2ADRB1ADRB3KCNH2KDM4E
SCHEMBL2019519 0.89 ADRB2 (0.72) ADRB2ADRB1ADRB3KCNH2KDM4E
SCHEMBL2019517 0.89 ADRB2 (0.72) ADRB2ADRB1ADRB3KCNH2KDM4E
SCHEMBL2022251 0.87 KCNH2 (0.78) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL2022248 0.87 KCNH2 (0.78) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL2022249 0.87 KCNH2 (0.78) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL2020741 0.86 ADRB2 (0.92) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL2020739 0.86 ADRB2 (0.92) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL2020737 0.86 ADRB2 (0.92) ADRB2ADRB1ADRB3KCNH2MAPT
SCHEMBL8781535 0.84 ADRB2 (1.00) ADRB2ADRB1ADRB3KCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994459-A Aryloxypropane substituted piperazine derivatives with antiarrhythmic and antifibrillatory activity AMERICAN HOME PRODUCTS CORPORATION (US) 1991-02-19 US disclosed