SCHEMBL9868540

SCHEMBL9868540

CCOn1nnc2cc(Cc3ccccc3-n3ccnc3)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
FGFR1 P11362 1/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
CYP19A1 P11511 1/20 0.35
IDO1 P14902 1/20 0.34
HTR5A P47898 1/20 0.34
KMT2A Q03164 7/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
MAPT P10636 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526934 0.88 FGFR1 (0.35) TSHRNPSR1RXFP1FGFR1CYP11B1
SCHEMBL3279905 0.82 CTNNB1 (0.46) FGFR1CYP11B1CYP11B2CYP19A1IDO1
SCHEMBL9869542 0.81 SLC9A1 (0.47) FGFR1IDO1HTR5APOLBMCHR1
SCHEMBL9524640 0.78 SLC9A1 (0.38) FGFR1CYP11B1CYP11B2CYP19A1IDO1
Nitric Acid SCHEMBL9527186 0.77 NSD2 (0.39) RXFP1IDO1KMT2ANPC1RAB9A
SCHEMBL7463718 0.76 NPC1 (0.44) FGFR1CYP11B1CYP11B2IDO1HTR5A
SCHEMBL3279244 0.75 IDO1 (0.41) NPSR1FGFR1CYP11B1CYP11B2CYP19A1
SCHEMBL9664804 0.74 CYP11B1 (0.40) TSHRNPSR1FGFR1CYP11B1CYP11B2
SCHEMBL9196161 0.74 IDO1 (0.43) NPSR1FGFR1CYP11B1CYP11B2CYP19A1
SCHEMBL9078567 0.72 FGFR1 (0.41) NPSR1FGFR1CYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5039677-A Estrogen inhibitor JANSSEN PHARMACEUTICA N.V. (CA) 1991-08-13 US disclosed
US-4943574-A AROMATASE INHIBITORS, ESTROGEN DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-24 US disclosed