SCHEMBL9869145

SCHEMBL9869145

COc1cc(N)c([N+](=O)[O-])cc1C(=O)NC1CCN(CCCc2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.60
CYP3A4 P08684 2/20 0.60
DRD2 P14416 2/20 0.60
ADRA2B P18089 2/20 0.60
ADRA2C P18825 2/20 0.60
SLC6A2 P23975 2/20 0.60
HTR2A P28223 2/20 0.60
DRD3 P35462 2/20 0.60
OPRK1 P41145 2/20 0.60
HTR2B P41595 2/20 0.60
CHRNA4 P43681 2/20 0.60
HTR3A P46098 2/20 0.60
SLC6A3 Q01959 2/20 0.60
KCNH2 Q12809 2/20 0.60
CYP1A2 P05177 1/20 0.60
ADRA2A P08913 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
ACHE P22303 1/20 0.60
HTR2C P28335 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867490 0.95 DRD4 (0.62) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9866244 0.90 DRD4 (0.75) DRD4CYP3A4DRD2ADRA2BADRA2C
Hydrochloric Acid SCHEMBL9867297 0.89 DRD4 (0.74) DRD4CYP3A4DRD2ADRA2BADRA2C
Iodomethane SCHEMBL9866905 0.88 DRD4 (0.73) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9866907 0.88 DRD4 (0.53) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9865657 0.83 DRD4 (0.63) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9866636 0.82 MCHR1 (0.59) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9866643 0.82 MCHR1 (0.59) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9867393 0.82 MCHR1 (0.62) DRD4CYP3A4DRD2ADRA2BADRA2C
SCHEMBL9866982 0.82 HTR4 (0.53) DRD2ADRA2BADRA2CSLC6A2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026858-A Used for treating nausea, vomating, gastrointestinal disorders and centarl nervous system WALTON S.A. (ES) 1991-06-25 US disclosed