SCHEMBL9870883

SCHEMBL9870883

O=C(O)c1cn(-c2ccc(F)cc2F)c2c(F)c(N3CCNCC3)c(F)cc2c1=O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 7/20 0.61
TOP1 P11387 4/20 0.61
TOP2B Q02880 4/20 0.60
KDM4E B2RXH2 7/20 0.59
ALDH1A1 P00352 6/20 0.59
HPGD P15428 6/20 0.59
HSD17B10 Q99714 6/20 0.59
LMNA P02545 4/20 0.59
POLB P06746 1/20 0.53
HSP90AA1 P07900 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
BRD4 O60885 1/20 0.52
TSHR P16473 1/20 0.52
HTT P42858 1/20 0.52
CYP2J2 P51589 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
KMT2A Q03164 2/20 0.49
PMP22 Q01453 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10702973 0.96 TOP2A (0.58) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL9870380 0.91 KDM4E (0.64) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL10769256 0.90 TOP2A (0.59) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL9773828 0.90 TOP2A (0.57) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL9662901 0.90 TOP2A (0.59) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL9871193 0.89 KDM4E (0.64) TOP2ATOP1KDM4EALDH1A1HPGD
SCHEMBL9662381 0.89 TOP2A (0.56) TOP2ATOP1TOP2BKDM4EALDH1A1
Hydrochloric Acid SCHEMBL9773735 0.88 TOP2A (0.55) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL9870203 0.88 KDM4E (0.66) TOP2ATOP1TOP2BKDM4EALDH1A1
SCHEMBL9869967 0.88 KDM4E (0.67) TOP2ATOP1TOP2BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4981854-A BACTERICIDES, ANIMAL GROWTH REGUALTORS BAYER AKTIENGESELLSCHAFT (DE) 1991-01-01 US disclosed
US-4980353-A BACTERICIDES, ANIMAL GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1990-12-25 US disclosed