SCHEMBL9870922

SCHEMBL9870922

C=CC(O)CC(O)CC(=O)OCC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
NR1I2 O75469 1/20 0.37
PGR P06401 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
PTGS2 P35354 1/20 0.37
PDE4D Q08499 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 4/20 0.36
TRPA1 O75762 1/20 0.36
TSHR P16473 3/20 0.35
ALOX15 P16050 4/20 0.35
CYP3A4 P08684 3/20 0.35
TDP1 Q9NUW8 2/20 0.35
KMT2A Q03164 2/20 0.35
HSD17B10 Q99714 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14283521 1.00 CYP1A2 (0.40) CYP1A2MGAMGAASIMGAM2
SCHEMBL6118705 0.85 GAA (0.44) CYP1A2MGAMGAASIMGAM2
SCHEMBL10773024 0.82 TSHR (0.46) GAAL3MBTL1ALDH1A1TSHRCYP3A4
SCHEMBL5497077 0.81 TSHR (0.39) MGAMGAASIMGAM2L3MBTL1
SCHEMBL14523084 0.81 TSHR (0.39) MGAMGAASIMGAM2L3MBTL1
SCHEMBL1258369 0.78 GAA (0.55) CYP1A2MGAMGAASIMGAM2
SCHEMBL12925787 0.78 GAA (0.41) CYP1A2MGAMGAASIMGAM2
SCHEMBL28172951 0.78 GAA (0.41) CYP1A2MGAMGAASIMGAM2
SCHEMBL15153932 0.77 L3MBTL1 (0.49) CYP1A2MGAMGAASIMGAM2
SCHEMBL2912543 0.77 MGAM (0.44) CYP1A2MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118772052-A Medical intermediate and preparation method thereof 湖南九维生物医药有限公司 2024-10-15 CN disclosed
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4957940-A ENZYME INHIBITORS, ANTILIPEMIC AGENTS WARNER-LAMBERT COMPANY (US) 1990-09-18 US disclosed
US-4950675-A ANTICHOLESTEROL AGENTS WARNER-LAMBERT COMPANY (US) 1990-08-21 US disclosed
US-4929620-A ANTILIPEMIC AGENTS WARNER-LAMBERT COMPANY (US) 1990-05-29 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
US-4906657-A Bicyclo heptane and bicyclo octane substituted inhibitors of cholesterol synthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
US-4868185-A HYPOLIPIDEMIC, ANTICHOLESTEROL WARNER-LAMBERT COMPANY (US) 1989-09-19 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed
US-4761419-A ANTILIPEMIC WARNER-LAMBERT COMPANY (US) 1988-08-02 US disclosed
US-4650890-A Preparation of olefinic compounds and intermediates thereof SANDOZ CORP. (US) 1987-03-17 US disclosed