SCHEMBL9871646

SCHEMBL9871646

Cn1c2c(c3ccccc31)C(=O)C(C(N)C1=NCCN1)CS2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 6/20 0.34
ADRA2B P18089 5/20 0.34
ADRA2C P18825 5/20 0.34
MYLK Q15746 2/20 0.33
NISCH Q9Y2I1 5/20 0.32
PRKD3 O94806 2/20 0.32
PRKCG P05129 2/20 0.32
PRKCB P05771 2/20 0.32
PRKCA P17252 2/20 0.32
PRKCH P24723 2/20 0.32
PRKCI P41743 2/20 0.32
PRKCE Q02156 2/20 0.32
PRKCQ Q04759 2/20 0.32
PRKCZ Q05513 2/20 0.32
PRKCD Q05655 2/20 0.32
PRKD1 Q15139 2/20 0.32
MAOA P21397 4/20 0.32
MAOB P27338 4/20 0.32
KCNH2 Q12809 3/20 0.32
CYP3A4 P08684 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871650 0.75 PRKD3 (0.40) ADRA2AADRA2BADRA2CPRKD3PRKCG
Hydrochloric Acid SCHEMBL9871784 0.71 ALDH1A1 (0.33) KCNH2CYP3A4CYP2D6
SCHEMBL9871149 0.70 CYP3A4 (0.38) PRKD3PRKCGPRKCBPRKCAPRKCH
Hydrochloric Acid SCHEMBL9872164 0.69 METAP1 (0.39) MYLKPRKD3PRKCGPRKCBPRKCA
SCHEMBL9872690 0.66 CYP3A4 (0.41) KCNH2CYP3A4CYP1A2CYP2D6HTR3E
SCHEMBL9870672 0.65 HDAC1 (0.42) KCNH2CYP3A4CYP1A2CYP2D6HTR3E
SCHEMBL9873374 0.65 PDGFRB (0.43) CYP2D6HTR2B
SCHEMBL9872923 0.65 KCNH2 (0.40) KCNH2CYP3A4CYP1A2CYP2D6HTR3E
SCHEMBL9571779 0.65 KCNH2 (0.38) ADRA2CKCNH2CYP3A4CYP1A2CYP2D6
SCHEMBL9870845 0.64 CYP3A4 (0.39) PRKD3PRKCGPRKCBPRKCAPRKCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5030646-A Treatment of diseases resulting from disfunction of seretoninergic system ADIR ET COMPAGNIE (FR) 1991-07-09 US disclosed