SCHEMBL9871768

SCHEMBL9871768

Fc1ccc(C(c2ccncc2)c2ccc(F)c(F)c2)cc1F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.57
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
SLC6A3 Q01959 1/20 0.50
DPP4 P27487 2/20 0.43
CYP11B1 P15538 5/20 0.42
CYP11B2 P19099 5/20 0.42
CYP17A1 P05093 3/20 0.42
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
DPP8 Q6V1X1 1/20 0.37
ROCK2 O75116 1/20 0.35
CYP3A4 P08684 3/20 0.34
CYP2C19 P33261 1/20 0.34
NAMPT P43490 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C8 P10632 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6933110 0.84 CES2 (0.47) CYP19A1AKR1C3AKR1C2CES2CES1
Ammonia Solution, Strong SCHEMBL5999466 0.79 AKR1C3 (0.42) CYP19A1SLC6A2SLC6A4SLC6A3DPP4
SCHEMBL29361168 0.76 SLC6A2 (0.78) CYP19A1SLC6A2SLC6A4SLC6A3CYP11B1
Ammonia Solution, Strong SCHEMBL6000329 0.74 CYP17A1 (0.58) CYP19A1SLC6A2SLC6A4SLC6A3DPP4
SCHEMBL11538836 0.73 CYP19A1 (1.00) CYP19A1SLC6A2SLC6A4SLC6A3CYP11B1
SCHEMBL940290 0.69 CYP19A1 (0.60) CYP19A1SLC6A2SLC6A4SLC6A3CYP11B1
SCHEMBL14242084 0.69 CYP19A1 (0.63) CYP19A1SLC6A2SLC6A4SLC6A3CYP11B1
SCHEMBL10460892 0.69 CYP19A1 (0.60) CYP19A1SLC6A2SLC6A4SLC6A3CYP11B1
SCHEMBL7440699 0.68 KMT2A (0.42) CYP19A1SLC6A2SLC6A4SLC6A3DPP4
SCHEMBL28193191 0.67 CES2 (0.45) AKR1C3AKR1C2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5057524-A Asthma, dermatitis A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US disclosed
US-4950674-A Arylalkylheterocyclic amines,N-substituted by aryloxyalkyl group in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1990-08-21 US disclosed