SCHEMBL9871905

SCHEMBL9871905

Oc1ccc(Cl)c2ccc(I)nc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.51
MAPT P10636 3/20 0.50
KDM4E B2RXH2 2/20 0.50
LMNA P02545 2/20 0.50
HSP90AA1 P07900 2/20 0.50
METAP2 P50579 2/20 0.50
METAP1 P53582 2/20 0.50
BRD4 O60885 1/20 0.50
OPRK1 P41145 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP3A4 P08684 3/20 0.35
MAPK1 P28482 2/20 0.35
ALDH1A1 P00352 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
TP53 P04637 1/20 0.34
APP P05067 1/20 0.34
CYP1A2 P05177 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3984759 0.80 MAPT (0.53) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL9062727 0.77 KMT2A (0.44) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL7692195 0.77 KMT2A (0.67) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL4293438 0.76 KMT2A (0.65) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL4286016 0.76 KMT2A (0.65) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL4304569 0.76 KMT2A (0.65) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL4393540 0.76 MAPT (0.49) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL4395732 0.76 MAPT (0.49) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL29154092 0.74 MAPT (0.46) PIM1MAPTKDM4ELMNAHSP90AA1
SCHEMBL1507963 0.73 MAPT (0.46) PIM1MAPTKDM4ELMNAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891627-B Ruthenium-containing coordination compound and preparation method thereof CHINESE ACAD INST CHEMISTRY 2015-04-29 CN claimed
CN-101891627-B Ruthenium-containing coordination compound and preparation method thereof CHINESE ACAD INST CHEMISTRY 2015-04-29 CN disclosed
US-5032402-A 3-hydroxy-N-methylpyrrolidone and use as transdermal enhancer THE UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1991-07-16 US disclosed
US-4973708-A TRANSDERMAL ENHANCER FOR PENETRATION OF DRUGS THROUGH THE SKIN UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1990-11-27 US disclosed