SCHEMBL9873088

SCHEMBL9873088

CCOc1nnc(OCC)c2c1nc(C1CCCCC1)n2Cc1ccc(-c2ccccc2C(=O)O)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 2/20 0.58
AGTR2 P50052 2/20 0.58
BRS3 P32247 1/20 0.45
PPARG P37231 4/20 0.44
ABCB11 O95342 1/20 0.44
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
CYP3A4 P08684 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CYP2C9 P11712 1/20 0.44
ADRB3 P13945 1/20 0.44
ADRA2B P18089 1/20 0.44
SLC6A2 P23975 1/20 0.44
TBXAS1 P24557 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
PDE3A Q14432 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9874436 0.92 AGTR1 (0.56) AGTR1AGTR2BRS3PPARG
SCHEMBL9873256 0.92 AGTR1 (0.56) AGTR1AGTR2BRS3PPARG
SCHEMBL9871651 0.90 AGTR1 (0.57) AGTR1AGTR2PPARG
SCHEMBL9874519 0.88 AGTR1 (0.56) AGTR1AGTR2BRS3PPARG
SCHEMBL9873489 0.88 AGTR1 (0.55) AGTR1AGTR2BRS3PPARG
SCHEMBL9873394 0.87 AGTR1 (0.55) AGTR1AGTR2BRS3PPARG
SCHEMBL9872455 0.87 AGTR1 (0.54) AGTR1AGTR2BRS3PPARG
SCHEMBL9874419 0.86 AGTR1 (0.54) AGTR1AGTR2BRS3
SCHEMBL9873902 0.86 AGTR1 (0.53) AGTR1AGTR2BRS3PPARG
SCHEMBL9872907 0.86 AGTR1 (0.53) AGTR1AGTR2BRS3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019715-A1 1H-SUBSTITUTED-IMIDAZO[4,5-d]PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-12-26 WO disclosed