SCHEMBL9873371

SCHEMBL9873371

Nc1c2c(nc3ccc(Cl)cc13)CCCC2=O

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 17/20 0.68
BCHE P06276 15/20 0.68
GRIN1 Q05586 10/20 0.68
GRIN2A Q12879 10/20 0.68
KDM4E B2RXH2 1/20 0.56
POLB P06746 1/20 0.51
RECQL P46063 1/20 0.51
CASP6 P55212 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
CHRM1 P11229 1/20 0.49
EPHX2 P34913 1/20 0.49
SLC2A1 P11166 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9876043 0.89 ACHE (0.63) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL9874322 0.86 ACHE (0.60) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL28984980 0.83 ACHE (0.66) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL10847043 0.83 ACHE (0.62) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL9068077 0.83 ACHE (0.66) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL10848027 0.83 ACHE (0.66) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL8006170 0.81 ACHE (1.00) ACHEBCHEGRIN1GRIN2ACHRM1
SCHEMBL10845002 0.80 KDM4E (0.53) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL10845569 0.80 ACHE (0.49) ACHEBCHEGRIN1GRIN2AKDM4E
SCHEMBL10848798 0.80 ACHE (0.67) ACHEBCHEGRIN1GRIN2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631286-A MEMORY ENHANCERS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-12-23 US claimed
EP-2681554-B1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON DICKINSON CO (US) 2017-08-09 EP disclosed
US-9459187-B2 Blood collection device containing lysophospholipase inhibitor BECTON, DICKINSON AND COMPANY (US) 2016-10-04 US disclosed
US-20140030754-A1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON, DICKINSON AND COMPANY (US) 2014-01-30 US disclosed
US-20130209985-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS BECTON, DICKINSON AND COMPANY 2013-08-15 US disclosed
EP-0179383-B1 9-AMINO-1,2,3,4-TETRAHYDROACRIDIN-1-OL AND RELATED COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-05-29 EP disclosed
US-4839364-A ALZHEIMER*S DISEASE; CHOLINESTERASE INHIBITORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-13 US disclosed
US-4835275-A Method of preparing 9-amino-1,2,3,4,-tetrahydroacridin-1-ones and related compounds HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-05-30 US disclosed
US-4754050-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-06-28 US disclosed
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
US-4631286-A MEMORY ENHANCERS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1986-12-23 US disclosed
EP-0179383-A2 9-Amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-04-30 EP disclosed