SCHEMBL9874235

SCHEMBL9874235

CCSc1ccnc(CSc2nc3ccccc3[nH]2)c1C

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.62
NPC1 O15118 8/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2D6 P10635 2/20 0.62
CYP2C9 P11712 2/20 0.62
CYP2C19 P33261 2/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2E1 P05181 1/20 0.53
CYP2C8 P10632 1/20 0.53
CYP2B6 P20813 1/20 0.53
NOS3 P29474 1/20 0.51
NOS1 P29475 1/20 0.51
NOS2 P35228 1/20 0.51
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 2/20 0.49
GALR3 O60755 1/20 0.49
MAPT P10636 1/20 0.49
STAT3 P40763 1/20 0.49
BCHE P06276 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9278218 0.91 RAB9A (0.60) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL10862355 0.90 RAB9A (0.52) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9278510 0.89 RAB9A (0.64) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9275547 0.88 RAB9A (0.66) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8412992 0.88 NPC1 (0.60) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914605 0.88 NPC1 (0.60) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL9279925 0.88 RAB9A (0.59) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL8914814 0.87 EPHX2 (0.61) RAB9ANPC1CYP1A2CYP2D6CYP2C9
SCHEMBL7812133 0.87 NPC1 (0.59) RAB9ANPC1CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8916118 0.87 RAB9A (0.56) RAB9ANPC1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0150586-B1 2-(PYRIDYLMETHYLTHIO)BENZIMIDAZOLES AND 2-(PYRIDYLMETHYLSULFINYL)BENZIMIDAZOLES THE UPJOHN COMPANY (US) 1991-05-08 EP claimed
EP-0150586-A2 2-(Pyridylmethylthio)benzimidazoles and 2-(pyridylmethylsulfinyl)benzimidazoles THE UPJOHN COMPANY (US) 1985-08-07 EP claimed
US-4873337-A N-substituted derivatives of 2-(pyridylalkenesulfinyl) benzimidazoles as gastric antisecretory agents THE UPJOHN COMPANY (US) 1989-10-10 US disclosed
EP-0176308-A2 2-(Pyridylalkylenesulfinyl) benzimidazoles THE UPJOHN COMPANY (US) 1986-04-02 EP disclosed