SCHEMBL9874579

SCHEMBL9874579

Cc1nc2c(OCc3ccccc3)nnc(O)c2n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 5/20 0.35
AGTR2 P50052 5/20 0.35
PDE3A Q14432 2/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE3B Q13370 1/20 0.35
ABCB11 O95342 1/20 0.34
EGFR P00533 1/20 0.34
ERBB2 P04626 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CYP2C9 P11712 1/20 0.34
ADRB3 P13945 1/20 0.34
ADRA2B P18089 1/20 0.34
SLC6A2 P23975 1/20 0.34
TBXAS1 P24557 1/20 0.34
HTR2C P28335 1/20 0.34
PPARG P37231 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9874827 0.93 AGTR1 (0.37) AGTR1AGTR2PDE3APDE4APDE4B
SCHEMBL9871494 0.90 PDE10A (0.36) AGTR1AGTR2PDE3AABCB11EGFR
SCHEMBL9874401 0.90 AGTR1 (0.36) AGTR1AGTR2PDE3AABCB11EGFR
SCHEMBL9873634 0.90 AGTR1 (0.37) AGTR1AGTR2PDE10A
SCHEMBL9873245 0.89 AGTR1 (0.34) AGTR1AGTR2PDE3APDE4APDE4B
SCHEMBL9873279 0.88 AGTR1 (0.34) AGTR1AGTR2
SCHEMBL9873895 0.87 AGTR1 (0.40) AGTR1AGTR2PDE10A
SCHEMBL9875077 0.87 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL9871582 0.87 AGTR1 (0.35) AGTR1AGTR2PPARGPDE10A
SCHEMBL9872857 0.86 AGTR1 (0.36) AGTR1AGTR2PDE3AABCB11EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019715-A1 1H-SUBSTITUTED-IMIDAZO[4,5-d]PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-12-26 WO disclosed