SCHEMBL9875491

SCHEMBL9875491

CC1=C(C(=O)O)C(c2ccccc2OC(F)F)C([N+](=O)[O-])=C(C)N1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.60
MAPT P10636 6/20 0.53
CYP1A2 P05177 6/20 0.53
ADORA3 P0DMS8 5/20 0.53
CYP2C9 P11712 5/20 0.53
CACNA1C Q13936 5/20 0.53
CYP3A4 P08684 4/20 0.53
CYP2C19 P33261 4/20 0.53
TSHR P16473 4/20 0.53
KMT2A Q03164 4/20 0.53
NFKB1 P19838 3/20 0.53
MEN1 O00255 3/20 0.53
CYP2D6 P10635 2/20 0.53
TP53 P04637 2/20 0.45
CACNA1B Q00975 4/20 0.44
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HPGD P15428 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
ABCC4 O15439 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875509 1.00 NR1I2 (0.60) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9875988 0.87 NR1I2 (0.61) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9874899 0.87 NR1I2 (0.61) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9806914 0.87 NR1I2 (0.76) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL10584053 0.86 NR1I2 (0.55) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL10517644 0.86 NR1I2 (0.54) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9875316 0.86 TSHR (0.62) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9874889 0.85 NR1I2 (0.58) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9875437 0.84 MAPT (0.58) NR1I2MAPTCYP1A2ADORA3CYP2C9
SCHEMBL9875432 0.84 MAPT (0.58) NR1I2MAPTCYP1A2ADORA3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008279-A Circulation-active fluoromethoxyphenyl dihydropyridine compounds BAYER AKTIENGESELLSCHAFT (DE) 1991-04-16 US disclosed
CN-1040192-A New fluorine methoxyphenyl dihydropyridine, its preparation method and the application aspect medicine BAYER AG (DE) 1990-03-07 CN disclosed
EP-0315018-A2 Fluoromethoxyphenyl-dihydropyridines, process for their preparation and their use in drugs BAYER AG (DE) 1989-05-10 EP disclosed
US-4764516-A Mixtures of optically active nitrodihydropyridines active on the circulatory system BAYER AKTIENGESELLSCHAFT (DE) 1988-08-16 US disclosed