SCHEMBL9875437

SCHEMBL9875437

CC1=C(C(=O)O)C(c2ccccc2OC(F)(F)F)C([N+](=O)[O-])=C(C)N1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.58
ADORA3 P0DMS8 6/20 0.58
CYP1A2 P05177 5/20 0.58
CACNA1C Q13936 5/20 0.58
CYP3A4 P08684 4/20 0.58
CYP2C9 P11712 4/20 0.58
CYP2C19 P33261 4/20 0.58
KMT2A Q03164 4/20 0.58
TSHR P16473 3/20 0.58
NFKB1 P19838 3/20 0.58
CYP2D6 P10635 2/20 0.58
MEN1 O00255 2/20 0.58
CACNA1B Q00975 4/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
ABCC4 O15439 2/20 0.44
CACNA1F O60840 2/20 0.44
ABCB11 O95342 2/20 0.44
LMNA P02545 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875432 1.00 MAPT (0.58) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL11009095 0.89 ADORA3 (0.74) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL9875554 0.86 MAPT (0.59) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL9875491 0.84 NR1I2 (0.60) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL9875509 0.84 NR1I2 (0.60) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL9875222 0.84 CACNA1C (0.56) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL9876069 0.83 CACNA1C (0.55) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL10408513 0.83 MAPT (0.78) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL4896908 0.83 MAPT (0.78) MAPTADORA3CYP1A2CACNA1CCYP3A4
SCHEMBL28830138 0.83 MAPT (0.78) MAPTADORA3CYP1A2CACNA1CCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008279-A Circulation-active fluoromethoxyphenyl dihydropyridine compounds BAYER AKTIENGESELLSCHAFT (DE) 1991-04-16 US disclosed