SCHEMBL9878296

SCHEMBL9878296

COc1cccc2c1C(=O)c1c(OC)cc(C)cc1C2=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 6/20 0.60
EGFR P00533 1/20 0.58
PIM1 P11309 1/20 0.58
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
ALDH1A1 P00352 4/20 0.54
MAPT P10636 3/20 0.54
CYP3A4 P08684 2/20 0.54
KDM4E B2RXH2 1/20 0.54
USP2 O75604 1/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
BRCA1 P38398 1/20 0.54
RECQL P46063 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
APAF1 O14727 1/20 0.54
MITF O75030 1/20 0.54
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
CYP1A2 P05177 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8930315 0.88 MAPT (0.73) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL16226264 0.88 ELANE (0.73) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL8947495 0.86 EGFR (0.73) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL26187210 0.83 ELANE (0.61) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL8996346 0.83 EGFR (0.56) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL30610014 0.83 ELANE (0.61) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL30040053 0.83 ELANE (0.61) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL15413483 0.83 EGFR (0.56) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL16226501 0.81 ELANE (0.61) ELANEEGFRPIM1MEN1KMT2A
SCHEMBL3417492 0.80 EGFR (0.76) ELANEEGFRPIM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5053431-A Antitumor-anticarcinogenic agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1991-10-01 US disclosed
US-4966918-A ANTICARCINOGENIC AGENTS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-10-30 US disclosed
WO-1990008759-A1 DERIVATIVES OF CHRYSOPHANOL SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-08-09 WO disclosed