SCHEMBL9878787

SCHEMBL9878787

Oc1nc(COCc2ccccc2)nc2c1SCCC2

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 11/20 0.38
PDE4D Q08499 11/20 0.38
TSHR P16473 2/20 0.38
KDM4E B2RXH2 3/20 0.32
POLB P06746 2/20 0.32
ALDH1A1 P00352 3/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
CA1 P00915 1/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878241 0.85 TSHR (0.38) PDE4BPDE4DTSHRALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL9877821 0.77 HTR2C (0.44)
Hydrochloric Acid SCHEMBL9877620 0.77 HTR2C (0.44)
SCHEMBL11108193 0.64 KDM4E (0.39) KDM4EALDH1A1L3MBTL1TP53MAPT
Cyclohexane SCHEMBL8149682 0.63 TSHR (0.83) TSHRKDM4EPOLBCA1LMNA
SCHEMBL14811521 0.63 TSHR (0.46) TSHRKDM4EPOLBALDH1A1L3MBTL1
Hydrogen Peroxide SCHEMBL28758135 0.63 TSHR (0.94) TSHRKDM4EPOLBALDH1A1L3MBTL1
Phenol SCHEMBL5486172 0.62 TSHR (0.79) TSHRKDM4EPOLBALDH1A1L3MBTL1
Phenol SCHEMBL21518644 0.62 TSHR (0.79) TSHRKDM4EPOLBALDH1A1L3MBTL1
Hydroquinone SCHEMBL51561 0.62 TSHR (0.79) TSHRKDM4EPOLBALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994464-A Treatment of elevated intraocular pressure and glaucoma MERCK & CO., INC. (US) 1991-02-19 US disclosed
US-4889856-A INTRAOCULAR PRESSURE REDUCTION; CARDIOVASCULAR DISORDERS MERCK & CO., INC. (US) 1989-12-26 US disclosed
EP-0276057-A2 Piperazinylpyrimidines as beta-adrenergic receptor blocking agents MERCK & CO. INC. (US) 1988-07-27 EP disclosed