SCHEMBL9892352

SCHEMBL9892352

CC(C)(C)C(=O)Nc1nc(C2CC2)cs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 1.00
TMIGD3 P0DMS9 3/20 1.00
TYR P14679 1/20 0.51
LMNA P02545 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HTT P42858 1/20 0.51
ADORA2A P29274 2/20 0.50
SMN1; SMN2 Q16637 5/20 0.49
MAPT P10636 4/20 0.49
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
NFKB1 P19838 2/20 0.49
NFKB2 Q00653 2/20 0.49
RELA Q04206 2/20 0.49
CCR2 P41597 1/20 0.48
ALDH1A1 P00352 3/20 0.48
TP53 P04637 1/20 0.48
FPR1 P21462 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ATAD2 Q6PL18 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9891514 0.93 ADORA1 (0.86) ADORA1TMIGD3TYRLMNAKDM4E
SCHEMBL16480470 0.83 ADORA1 (0.70) ADORA1TMIGD3TYRLMNAKDM4E
SCHEMBL4304336 0.81 ADORA1 (0.68) ADORA1TMIGD3ADORA2ASMN1; SMN2MAPT
SCHEMBL4969168 0.81 ADORA1 (0.68) ADORA1TMIGD3LMNAADORA2ASMN1; SMN2
SCHEMBL9891909 0.79 ADORA1 (0.65) ADORA1TMIGD3TYRLMNAADORA2A
SCHEMBL9893165 0.79 ADORA1 (0.65) ADORA1TMIGD3LMNAKDM4EADORA2A
SCHEMBL3784705 0.79 ADORA1 (0.64) ADORA1TMIGD3TYRLMNAKDM4E
SCHEMBL16358870 0.78 ADORA1 (0.62) ADORA1TMIGD3ADORA2ASMN1; SMN2MAPT
SCHEMBL1464818 0.78 ADORA1 (0.62) ADORA1TMIGD3LMNAKDM4EHTT
SCHEMBL15219031 0.77 ADORA1 (0.61) ADORA1TMIGD3ADORA2ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120142677-A1 Pyrrolidine Compounds Which Modulate The CB2 Receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142677-A1 Pyrrolidine Compounds Which Modulate The CB2 Receptor CNR2, CNR1, OPRL1 ADORA1 278/4885TMIGD3 1180/4885TYR 2678/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.