SCHEMBL989896

SCHEMBL989896

COc1ccc(C=O)cc1-c1cc(F)cc(C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.45
TSHR P16473 1/20 0.45
ERN1 O75460 2/20 0.44
AOX1 Q06278 1/20 0.42
HPGD P15428 2/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
FDPS P14324 1/20 0.40
KDM1A O60341 1/20 0.40
EPAS1 Q99814 1/20 0.39
TRIM24 O15164 1/20 0.39
ALDH5A1 P51649 1/20 0.39
ABAT P80404 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TRIM33 Q9UPN9 1/20 0.39
TTR P02766 1/20 0.38
PGR P06401 2/20 0.38
AR P10275 1/20 0.38
AGPAT2 O15120 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8433481 0.82 ALDH1A1 (0.51) ALDH1A1TSHRAOX1HPGDFDPS
SCHEMBL1812724 0.82 ALDH1A1 (0.47) ALDH1A1TSHRAOX1HPGDFDPS
SCHEMBL988687 0.80 KDM4E (0.41) ALDH1A1HPGDKDM1ATRIM24ALDH5A1
SCHEMBL1077197 0.79 PTGDR2 (0.41) ALDH1A1POLBEPAS1AR
SCHEMBL3924578 0.78 ALDH1A1 (0.56) ALDH1A1TSHRERN1AOX1HPGD
SCHEMBL16180046 0.76 KDM1A (0.47) ALDH1A1TSHRAOX1KDM1ATTR
SCHEMBL16711689 0.73 ALDH1A1 (0.58) ALDH1A1TSHRERN1AOX1HPGD
SCHEMBL24028315 0.72 ALDH1A1 (0.53) ALDH1A1TSHRERN1AOX1HPGD
SCHEMBL17969078 0.72 ALDH1A1 (0.53) ALDH1A1TSHRERN1AOX1HPGD
SCHEMBL2002821 0.72 ERN1 (0.59) ALDH1A1TSHRERN1AOX1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002814-A2 BIARYL OXYACETIC ACID COMPOUNDS LIGAND PHARMACEUTICALS INC. (US) 2011-01-06 WO disclosed
WO-2011002814-A2 BIARYL OXYACETIC ACID COMPOUNDS LIGAND PHARMACEUTICALS INC. (US) 2011-01-06 WO disclosed