SCHEMBL9901190

SCHEMBL9901190

CCOC(=O)c1nc2cscc2nc1C(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
CYP1A2 P05177 3/20 0.40
GLP1R P43220 1/20 0.40
SLC10A2 Q12908 1/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 3/20 0.37
MAPK1 P28482 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
GAA P10253 2/20 0.37
HPGD P15428 1/20 0.37
ATM Q13315 1/20 0.37
TARBP2 Q15633 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21177166 0.70 BRD4 (0.47) ALDH1A1CYP1A2NPC1MAPTKDM4E
SCHEMBL30040951 0.68 KDM4E (0.51) ALDH1A1CYP1A2KMT2ANPC1MEN1
SCHEMBL22213904 0.68 HTT (0.47) ALDH1A1CYP1A2KMT2AMEN1MAPT
SCHEMBL15614506 0.68 KDM4E (0.40) ALDH1A1CYP1A2KMT2ANPC1MEN1
SCHEMBL1498218 0.66 TSHR (0.59) ALDH1A1CYP1A2KMT2ANPC1MEN1
SCHEMBL4294216 0.66 KMT2A (0.46) ALDH1A1KMT2ANPC1MEN1MAPT
SCHEMBL28979284 0.66 GAA (0.52) ALDH1A1CYP1A2KMT2ANPC1MEN1
SCHEMBL7233421 0.66 NPC1 (0.54) ALDH1A1CYP1A2KMT2ANPC1MEN1
SCHEMBL1431368 0.66 ALDH1A1 (0.47) ALDH1A1CYP1A2KMT2ANPC1MEN1
SCHEMBL166847 0.66 SMN1; SMN2 (0.46) ALDH1A1CYP1A2KMT2ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076966-A1 SUBSTITUTED THIENO [3,4-B] PYRAZINE COMPOUNDS LUPIN LIMITED (IN) 2012-06-14 WO disclosed
WO-2012076966-A1 SUBSTITUTED THIENO [3,4-B] PYRAZINE COMPOUNDS LUPIN LIMITED (IN) 2012-06-14 WO disclosed