SCHEMBL9901547

SCHEMBL9901547

CS(=O)(=O)OCc1nc([C]2CC2)co1

nearest known ligand 0.30

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9901549 0.77 SCN5A (0.33)
SCHEMBL1166849 0.72 CYP1A2 (0.38) CYP1A2CYP3A4CYP2D6
SCHEMBL856703 0.71 CYP1A2 (0.30) CYP1A2CYP3A4CYP2D6
SCHEMBL9900516 0.70 CYP1A2 (0.31) CYP1A2CYP3A4CYP2D6
SCHEMBL1707146 0.68 CYP1A2 (0.43) CYP1A2
SCHEMBL1166447 0.65
SCHEMBL1161169 0.65 KDM4E (0.31) CYP1A2CYP3A4CYP2D6
SCHEMBL4031429 0.64 DAO (0.35) CYP1A2CYP3A4CYP2D6
SCHEMBL3086180 0.62 CYP1A2 (0.32) CYP1A2CYP3A4CYP2D6
SCHEMBL16828409 0.61 MAPT (0.51) CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648724-A1 HYDROXYLATED AMINOTRIAZOLE DERIVATIVES AS ALX RECEPTOR AGONISTS Actelion Pharmaceuticals Ltd. (CH) 2013-10-16 EP disclosed
WO-2012077051-A1 HYDROXYLATED AMINOTRIAZOLE DERIVATIVES AS ALX RECEPTOR AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2012-06-14 WO disclosed