SCHEMBL9901805

SCHEMBL9901805

Cc1cc(CNC(=O)c2nc3n(c(=O)c2O)CC2(F)CC[C]3CC2)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 9/20 0.44
KCNH2 Q12809 1/20 0.39
CYP2C9 P11712 1/20 0.39
MMP10 P09238 4/20 0.38
MMP8 P22894 4/20 0.38
MMP9 P14780 1/20 0.37
SCD O00767 1/20 0.37
KCNE1 P15382 1/20 0.36
CCR1 P32246 1/20 0.36
KCNQ1 P51787 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MYC P01106 1/20 0.35
WDR5 P61964 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904944 0.83 MMP13 (0.39) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL9904932 0.83 MMP13 (0.39) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL9904934 0.83 MMP13 (0.36) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL9901158 0.82 CYP2C9 (0.44) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL52487 0.80 KCNH2 (0.48) KCNH2CYP2C9KCNE1CCR1KCNQ1
SCHEMBL9901256 0.80 CYP2C9 (0.42) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL9904978 0.80 MMP13 (0.36) MMP13KCNH2CYP2C9SCDWDR5
SCHEMBL9901113 0.80 KCNH2 (0.38) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL9905205 0.79 MMP13 (0.39) MMP13KCNH2CYP2C9MMP10MMP8
SCHEMBL9901114 0.79 KCNH2 (0.37) MMP13KCNH2CYP2C9MMP10MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649077-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP claimed
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO claimed
EP-2649077-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP disclosed
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed