SCHEMBL9903015

SCHEMBL9903015

N#Cc1cccc(C(C(c2cccnc2)c2cccnc2)n2ccccc2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.41
MGLL Q99685 1/20 0.41
VNN1 O95497 1/20 0.39
KCNA5 P22460 4/20 0.39
KCNH2 Q12809 2/20 0.39
CREBBP Q92793 1/20 0.39
CYP11B1 P15538 4/20 0.37
CYP11B2 P19099 4/20 0.37
CHRNB2 P17787 2/20 0.35
CHRNA5 P30532 2/20 0.35
CHRNA4 P43681 2/20 0.35
TNF P01375 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
SGMS2 Q8NHU3 1/20 0.34
CYP17A1 P05093 1/20 0.34
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1242156 0.84 CFTR (0.42) CYP19A1KCNA5CREBBPCYP11B1CYP11B2
SCHEMBL1242972 0.78 KCNA5 (0.46) CYP19A1MGLLVNN1KCNA5KCNH2
SCHEMBL1242330 0.77 MGLL (0.46) CYP19A1MGLLVNN1KCNA5KCNH2
SCHEMBL1242145 0.77 CYP19A1 (0.45) CYP19A1MGLLVNN1KCNA5KCNH2
SCHEMBL1242623 0.76 KCNA5 (0.44) CYP19A1KCNA5CYP11B1CYP11B2GAA
SCHEMBL1243093 0.76 MGLL (0.42) CYP19A1MGLLVNN1KCNA5KCNH2
SCHEMBL1242929 0.76 KCNA5 (0.40) CYP19A1MGLLVNN1KCNA5KCNH2
SCHEMBL1378201 0.75 CYP19A1 (0.51) CYP19A1MGLLVNN1KCNA5KCNH2
SCHEMBL1243310 0.75 KCNA5 (0.40) KCNA5KCNH2ALDH1A1
SCHEMBL1241967 0.75 KCNA5 (0.40) KCNA5KCNH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781635-B1 POTASSIUM CHANNEL INHIBITORS MERCK SHARP & DOHME (US) 2012-06-13 EP claimed