SCHEMBL9909370

SCHEMBL9909370

Cc1cccc(C(Cc2ccc(C)c(C)c2)c2ccc(CO)cc2Br)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.36
CTSB P07858 3/20 0.34
PSMB8 P28062 2/20 0.33
PSMB5 P28074 2/20 0.33
ACP3 P15309 1/20 0.32
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31
THRA P10827 1/20 0.31
THRB P10828 1/20 0.31
CYP19A1 P11511 1/20 0.30
NR3C2 P08235 1/20 0.30
CTSL P07711 1/20 0.30
CTSS P25774 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9909383 0.80 CETP (0.35) S1PR1CTSBGAA
SCHEMBL9909371 0.79 CTSA (0.34) S1PR1CTSBPSMB8PSMB5GAA
SCHEMBL9112164 0.77 CTSB (0.32) S1PR1CTSB
SCHEMBL9104789 0.70 CTSB (0.44) CTSBPSMB8PSMB5ACP3CTSL
SCHEMBL9909373 0.69 S1PR1 (0.54) S1PR1ACP3
SCHEMBL93048 0.67 S1PR1 (0.47) S1PR1GAA
SCHEMBL10060821 0.67 S1PR1 (0.51) S1PR1
SCHEMBL9909384 0.67 S1PR1 (0.53) S1PR1CTSBPSMB8PSMB5
SCHEMBL9110842 0.66 ESR1 (0.41) CTSBPSMB8PSMB5ACP3GAA
SCHEMBL1467659 0.66 HPGD (0.42) S1PR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120142640-A1 ALKYNE AND ALKENE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE-1 RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-07 US disclosed
WO-2012074921-A1 ALKYNE AND ALKENE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE-1 RECEPTOR MODULATORS ALLERGAN, INC. (US) 2012-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142640-A1 ALKYNE AND ALKENE DERIVATIVES AS SPHINGOSINE 1-PHOSPHATE-1 RECEPTOR MODULATORS S1PR1, S1PR3, S1PR2 S1PR1 1/4885CTSB 2311/4885PSMB8 4211/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.