SCHEMBL9911541

SCHEMBL9911541

CC(C)C(=O)Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.55
MEN1 O00255 3/20 0.55
CYP2C19 P33261 2/20 0.54
CYP1A2 P05177 1/20 0.54
TSHR P16473 1/20 0.52
MAPT P10636 4/20 0.51
GAA P10253 1/20 0.51
PKM P14618 1/20 0.51
ALDH1A1 P00352 5/20 0.50
LOXL2 Q9Y4K0 1/20 0.50
HTT P42858 2/20 0.49
MAPK1 P28482 1/20 0.48
LMNA P02545 1/20 0.48
THRB P10828 1/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008660 0.84 TSHR (0.56) KMT2AMEN1CYP2C19TSHRMAPT
SCHEMBL13197240 0.84 POLB (0.45) CYP1A2TSHRGAAALDH1A1HTT
SCHEMBL29318769 0.82 TSHR (0.53) KMT2ACYP2C19TSHRMAPTALDH1A1
SCHEMBL7733270 0.81 CYP2C19 (0.57) KMT2AMEN1CYP2C19CYP1A2TSHR
SCHEMBL43494 0.81 CYP2C19 (0.57) KMT2AMEN1CYP2C19CYP1A2TSHR
SCHEMBL6932662 0.80 CYP2C19 (0.61) KMT2AMEN1CYP2C19CYP1A2TSHR
SCHEMBL9911538 0.80 TSHR (0.56) CYP2C19CYP1A2TSHRALDH1A1HTT
SCHEMBL1625876 0.79 MEN1 (0.56) KMT2AMEN1CYP2C19CYP1A2TSHR
SCHEMBL1625595 0.79 MEN1 (0.56) KMT2AMEN1CYP2C19CYP1A2TSHR
SCHEMBL1625885 0.79 MEN1 (0.56) KMT2AMEN1CYP2C19CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9745280-B2 Compound or pharmaceutically acceptable salt thereof, and pharmaceutical composition containing same as active ingredient SNU R&DB FOUNDATION (KR) 2017-08-29 US disclosed
US-9745280-B2 Compound or pharmaceutically acceptable salt thereof, and pharmaceutical composition containing same as active ingredient SNU R&DB FOUNDATION (KR) 2017-08-29 US disclosed
US-9562186-B2 Oligomeric and polymeric electronically-modified boronic acids and methods of using the same HALLIBURTON ENERGY SERVICES, INC. (US) 2017-02-07 US disclosed
US-20160340331-A1 NOVEL COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT SNU R&DB FOUNDATION (KR) 2016-11-24 US disclosed
US-20150210918-A1 OLIGOMERIC AND POLYMERIC ELECTRONICALLY-MODIFIED BORONIC ACIDS AND METHODS OF USING THE SAME HALLIBURTON ENERGY SERVICES, INC. (US) 2015-07-30 US disclosed
US-9057698-B2 Methods of chemoselective derivation of multiple classes of metabolites BROWN UNIVERSITY (US) 2015-06-16 US disclosed
US-9027644-B2 Oligomeric and polymeric electronically-modified boronic acids and methods of using the same HALLIBURTON ENERGY SERVICES, INC. (US) 2015-05-12 US disclosed
US-20140174748-A1 OLIGOMERIC AND POLYMERIC ELECTRONICALLY-MODIFIED BORONIC ACIDS AND METHODS OF USING THE SAME HALLIBURTON ENERGY SERVICES, INC. (US) 2014-06-26 US disclosed
US-20140110120-A1 Oligomeric and Polymeric Electronically-Modified Boronic Acids and Methods of Using the Same HALLIBURTON ENERGY SERVICES, INC. (US) 2014-04-24 US disclosed
US-20130071940-A1 METHODS OF CHEMOSELECTIVE DERIVATION OF MULTIPLE CLASSES OF METABOLITES BROWN UNIVERSITY (US) 2013-03-21 US disclosed
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-7517998-B2 Benzothiazole or benzothiazine derivative of dipyrido(2,3;b:2',3'-e) diazepin-6-one; viricide against human t-cell leukemia/lymphoma virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2009-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160340331-A1 NOVEL COMPOUND OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING SAME AS ACTIVE INGREDIENT HSP90AB1, HSP90AA1, HSP90AB2P KMT2A 3179/4885MEN1 4632/4885CYP2C19 3149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.