SCHEMBL9912199

SCHEMBL9912199

O=c1ccc(-c2cc(NCCc3c(F)cccc3Cl)nc(O)n2)c[nH]1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGDR Q13258 5/20 0.51
LCK P06239 3/20 0.37
BTK Q06187 3/20 0.37
MAPK14 Q16539 2/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
CNR1 P21554 1/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
DAO P14920 2/20 0.36
ALDH2 P05091 1/20 0.35
CD38 P28907 1/20 0.35
AKR1B1 P15121 1/20 0.34
RAB9A P51151 2/20 0.34
TAAR1 Q96RJ0 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4500166 0.86 PTGDR (0.51) PTGDRLCKBTKROCK2ROCK1
SCHEMBL4501709 0.86 PTGDR (0.70) PTGDR
SCHEMBL9912207 0.78 PTGDR (0.51) PTGDRLCKBTKMAPK14CNR1
SCHEMBL9912195 0.77 PTGDR (0.41) PTGDRMEN1KMT2A
SCHEMBL13895066 0.76 PTGDR (0.47) PTGDRLCKBTKMAPK14KDM4E
SCHEMBL14405092 0.75 PTGDR (0.41) PTGDRTP53
SCHEMBL4490256 0.72 PTGDR (0.75) PTGDRLCKBTKMAPK14
SCHEMBL10476050 0.70 PTGDR (0.47) PTGDRLCKBTKROCK2ROCK1
SCHEMBL4487437 0.70 PTGDR (0.74) PTGDR
SCHEMBL4503611 0.69 PTGDR (0.74) PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8193183-B2 2,6-substituted-4-monosubstitutedamino-pyrimidine as prostaglandin D2 receptor antagonists AVENTIS PHARMACEUTICALS INC. (US) 2012-06-05 US disclosed