SCHEMBL9912402

SCHEMBL9912402

CN/N=C(/C)Nc1ccc(C2CC2)cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.34
RAB9A P51151 4/20 0.34
NPC1 O15118 3/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPK14 Q16539 1/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
TP53 P04637 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
HTT P42858 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
SMURF2 Q9HAU4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9912470 0.83 NPC1 (0.36) JAK3RAB9ANPC1NFKB1NFKB2
SCHEMBL9912388 0.81 SLC6A2 (0.33) JAK3RAB9ANPC1NFKB1SLC6A2
SCHEMBL878961 0.79 CA1 (0.51) JAK3RAB9ANPC1MAPK14HTT
SCHEMBL1755259 0.77 RAB9A (0.48) RAB9ANPC1SMN1; SMN2TP53HTT
SCHEMBL9612039 0.75 SLC6A2 (0.35) RAB9ANPC1NFKB1SMN1; SMN2SLC6A2
SCHEMBL11407168 0.74 JAK3 (0.38) JAK3RAB9ANPC1NFKB1NFKB2
SCHEMBL11149788 0.73 HDAC3 (0.43) JAK3RAB9ANPC1CYP1A2HTT
SCHEMBL11283209 0.73 NPC1 (0.43) JAK3RAB9ANPC1NFKB1NFKB2
SCHEMBL11160172 0.73 JAK3 (0.37) JAK3RAB9ANPC1NFKB1NFKB2
SCHEMBL3824109 0.72 CA1 (0.48) JAK3RAB9ANPC1SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-7517998-B2 Benzothiazole or benzothiazine derivative of dipyrido(2,3;b:2',3'-e) diazepin-6-one; viricide against human t-cell leukemia/lymphoma virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2009-04-14 US disclosed