Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | ALDH1A1 | P00352 | 4/20 | 0.47 |
| ▸ | EPHX2 | P34913 | 1/20 | 0.41 |
| ▸ | TSHR | P16473 | 5/20 | 0.40 |
| ▸ | TDP1 | Q9NUW8 | 3/20 | 0.40 |
| ▸ | LMNA | P02545 | 2/20 | 0.40 |
| ▸ | NFKB1 | P19838 | 1/20 | 0.40 |
| ▸ | PMP22 | Q01453 | 1/20 | 0.40 |
| ▸ | CA12 | O43570 | 1/20 | 0.39 |
| ▸ | CA1 | P00915 | 1/20 | 0.39 |
| ▸ | CA2 | P00918 | 1/20 | 0.39 |
| ▸ | CA9 | Q16790 | 1/20 | 0.39 |
| ▸ | MAOA | P21397 | 1/20 | 0.39 |
| ▸ | MAOB | P27338 | 1/20 | 0.39 |
| ▸ | GPR84 | Q9NQS5 | 7/20 | 0.38 |
| ▸ | PPARG | P37231 | 6/20 | 0.38 |
| ▸ | PPARD | Q03181 | 6/20 | 0.38 |
| ▸ | PPARA | Q07869 | 6/20 | 0.38 |
| ▸ | HDAC11 | Q96DB2 | 5/20 | 0.38 |
| ▸ | TLR2 | O60603 | 2/20 | 0.38 |
| ▸ | MEN1 | O00255 | 2/20 | 0.38 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL3486013 | 1.00 | ALDH1A1 (0.47) | ALDH1A1EPHX2TSHRTDP1LMNA | |
| SCHEMBL5490052 | 1.00 | ALDH1A1 (0.47) | ALDH1A1EPHX2TSHRTDP1LMNA | |
| SCHEMBL7519278 | 0.88 | PAOX (0.42) | TDP1CA12CA1CA2CA9 | |
| SCHEMBL8374138 | 0.86 | MEN1 (0.39) | TDP1LMNACA12CA1CA2 | |
| SCHEMBL3485693 | 0.85 | TSHR (0.44) | ALDH1A1TSHRTDP1LMNACA12 | |
| SCHEMBL3486237 | 0.84 | TDP1 (0.43) | EPHX2TSHRTDP1LMNACA12 | |
| SCHEMBL15341460 | 0.83 | EPHX1 (0.46) | TDP1CA12CA1CA2CA9 | |
| SCHEMBL7527615 | 0.83 | EPHX1 (0.46) | TDP1CA12CA1CA2CA9 | |
| SCHEMBL5493650 | 0.83 | TDP1 (0.59) | TDP1CA12CA1CA2CA9 | |
| SCHEMBL5498803 | 0.83 | TDP1 (0.42) | TDP1CA12CA1CA2CA9 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20170114133-A1 | TEM8 ANTIBODIES AND METHODS OF USE | BIOMED VALLEY DISCOVERIES INC (US) | 2017-04-27 | — | — | US | disclosed |
| WO-2015191623-A1 | TEM8 ANTIBODIES AND METHODS OF USE | BIOMED VALLEY DISCOVERIES, INC. (US) | 2015-12-17 | — | — | WO | disclosed |
| US-20140065172-A1 | DELIVERY SYSTEM AND CONJUGATES FOR COMPOUND DELIVERY VIA NATURALLY OCCURRING INTRACELLULAR TRANSPORT ROUTES | ARROWHEAD RESEARCH CORPORATION | 2014-03-06 | — | — | US | disclosed |
| EP-2667898-A1 | DELIVERY SYSTEM AND CONJUGATES FOR COMPOUND DELIVERY VIA NATURALLY OCCURRING INTRACELLULAR TRANSPORT ROUTES | Cenix Bioscience GmbH (DE) | 2013-12-04 | — | — | EP | disclosed |
| US-20120258104-A1 | Delivery System and Conjugates For Compound Delivery Via Naturally Occurring Intracellular Transport Routes | CENIX BIOSCIENCE GMBH (DE) | 2012-10-11 | — | — | US | disclosed |
| WO-2012101235-A1 | DELIVERY SYSTEM AND CONJUGATES FOR COMPOUND DELIVERY VIA NATURALLY OCCURRING INTRACELLULAR TRANSPORT ROUTES | CENIX BIOSCIENCE GMBH (DE) | 2012-08-02 | — | — | WO | disclosed |
| EP-2456470-A1 | DELIVERY SYSTEM AND CONJUGATES FOR COMPOUND DELIVERY VIA NATURALLY OCCURRING INTRACELLULAR TRANSPORT ROUTES | Cenix Bioscience GmbH (DE) | 2012-05-30 | — | — | EP | disclosed |
| WO-2011009624-A1 | DELIVERY SYSTEM AND CONJUGATES FOR COMPOUND DELIVERY VIA NATURALLY OCCURRING INTRACELLULAR TRANSPORT ROUTES | CENIX BIOSCIENCE GMBH (DE) | 2011-01-27 | — | — | WO | disclosed |