SCHEMBL992204

SCHEMBL992204

C=CCC(Oc1cccc(Cl)c1C)N1CCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.38
SLC6A3 Q01959 2/20 0.38
SLC6A4 P31645 1/20 0.38
HTR7 P34969 2/20 0.37
HTR6 P50406 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HSD11B1 P28845 3/20 0.34
NR1I2 O75469 1/20 0.34
TSHR P16473 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1079194 0.81 HTR7 (0.39) HTR7HTR6SMN1; SMN2ALDH1A1HSD11B1
SCHEMBL1079190 0.81 HTR7 (0.39) HTR7HTR6SMN1; SMN2ALDH1A1HSD11B1
SCHEMBL991769 0.80 HTR7 (0.39) SLC6A2SLC6A3SLC6A4HTR7HTR6
SCHEMBL11539874 0.71 TSHR (0.44) SLC6A2SLC6A3SLC6A4HTR7HTR6
SCHEMBL11538270 0.70 TSHR (0.47) SLC6A2SLC6A3SLC6A4HTR7HTR6
SCHEMBL20041877 0.69 SLC6A4 (0.45) SLC6A2SLC6A3SLC6A4HTR6CYP2D6
SCHEMBL1060453 0.68 SLC6A4 (0.46) SLC6A2SLC6A3SLC6A4CYP2D6
SCHEMBL1060452 0.68 SLC6A4 (0.46) SLC6A2SLC6A3SLC6A4CYP2D6
SCHEMBL1079151 0.68 HTR7 (0.54) SLC6A2SLC6A3SLC6A4HTR7HTR6
SCHEMBL1079153 0.68 HTR7 (0.54) SLC6A2SLC6A3SLC6A4HTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2454234-A2 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS Theravance, Inc. (US) 2012-05-23 EP disclosed
WO-2011008666-A2 3-PHENOXYMETHYLPYRROLIDINE COMPOUNDS THERAVANCE, INC. (US) 2011-01-20 WO disclosed