SCHEMBL9923381

SCHEMBL9923381

Cc1cnc2[nH]cc(C#N)c2c1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 7/20 0.45
CDC42BPB Q9Y5S2 7/20 0.43
ROCK2 O75116 6/20 0.43
ROCK1 Q13464 6/20 0.43
CDC42BPA Q5VT25 3/20 0.43
HSP90AB1 P08238 1/20 0.42
MAP3K7 O43318 1/20 0.39
TAB1 Q15750 1/20 0.39
CHUK O15111 2/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
JAK3 P52333 1/20 0.38
MAP3K5 Q99683 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12590787 0.72 CHUK (0.48) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL26095838 0.70 ROCK2 (0.48) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL22026399 0.70 LRRK2 (0.46) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL16190651 0.69 LRRK2 (0.67) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL14649086 0.67 MAP3K7 (0.56) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL2600504 0.67 LRRK2 (0.39) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL29878823 0.67 KDM4E (0.41)
SCHEMBL20641160 0.67 LRRK2 (0.46) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL12590786 0.66 MAP3K7 (0.51) LRRK2CDC42BPBROCK2ROCK1CDC42BPA
SCHEMBL15758053 0.64 S1PR2 (0.42) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078802-A1 PREPARATION OF SUBSTITUTED-4,5-DIHYDROPYRROLO[4,3,2-de][2,6]NAPHTHYRIDIN-3(1H)-ONES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-06-14 WO disclosed