SCHEMBL9923446

SCHEMBL9923446

Cc1ccc(NC(=O)c2cc(Oc3ccc(C(=O)N4CCC4)c(C)c3)c3c(c2)OC(C)(CO)C3)nc1

nearest known ligand 0.87

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCK P35557 13/20 0.87
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
KCNH2 Q12809 6/20 0.43
MITF O75030 1/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
CNR1 P21554 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL645047 0.93 GCK (1.00) GCKNPC1RAB9AKCNH2MITF
SCHEMBL643901 0.83 GCK (0.66) GCKNPC1RAB9AKCNH2L3MBTL1
SCHEMBL645334 0.82 GCK (0.78) GCKNPC1RAB9AKCNH2MITF
SCHEMBL646447 0.81 GCK (0.75) GCKNPC1RAB9AKCNH2MITF
SCHEMBL643669 0.81 GCK (0.84) GCKKCNH2
SCHEMBL646229 0.79 GCK (0.74) GCKNPC1RAB9AKCNH2MITF
SCHEMBL644431 0.79 GCK (0.71) GCKNPC1RAB9AKCNH2MITF
SCHEMBL15780547 0.76 GCK (0.58) GCKNPC1RAB9AKCNH2L3MBTL1
SCHEMBL2644922 0.76 GCK (0.72) GCKNPC1GAACNR1
SCHEMBL643010 0.75 L3MBTL1 (0.57) GCKNPC1RAB9AKCNH2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed