SCHEMBL9923462

SCHEMBL9923462

CCOC(=O)c1cc(Oc2ccc(S)cc2)c2cc(C(=O)O)oc2c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.41
HPGD P15428 1/20 0.40
AKR1B1 P15121 1/20 0.39
ICAM1 P05362 1/20 0.39
SELE P16581 1/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 1/20 0.39
SLC2A1 P11166 1/20 0.39
THRA P10827 2/20 0.37
THRB P10828 2/20 0.37
GCK P35557 1/20 0.37
MAOB P27338 1/20 0.36
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10253338 0.91 PTGS2 (0.48) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL646057 0.86 PTGS2 (0.39) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL645021 0.86 GCK (0.49) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL12101428 0.84 HPGD (0.39) PTGS2HPGDICAM1SELEKDM4E
SCHEMBL2663647 0.84 PTGS2 (0.37) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL10253218 0.80 PTGS2 (0.47) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL12101423 0.76 SLC6A4 (0.42) PTGS2HPGDICAM1SELEALDH1A1
SCHEMBL643757 0.76 GCK (0.47) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL642524 0.76 GCK (0.41) PTGS2HPGDAKR1B1ICAM1SELE
SCHEMBL10257477 0.76 PTGS2 (0.48) PTGS2HPGDICAM1SELEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed