Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | MAPT | P10636 | 2/20 | 0.36 |
| ▸ | KDM4E | B2RXH2 | 3/20 | 0.36 |
| ▸ | GAA | P10253 | 3/20 | 0.36 |
| ▸ | RAB9A | P51151 | 1/20 | 0.36 |
| ▸ | MEN1 | O00255 | 1/20 | 0.33 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.33 |
| ▸ | HDAC1 | Q13547 | 7/20 | 0.33 |
| ▸ | HDAC3 | O15379 | 6/20 | 0.33 |
| ▸ | HDAC4 | P56524 | 6/20 | 0.33 |
| ▸ | HDAC7 | Q8WUI4 | 6/20 | 0.33 |
| ▸ | HDAC2 | Q92769 | 6/20 | 0.33 |
| ▸ | HDAC11 | Q96DB2 | 6/20 | 0.33 |
| ▸ | HDAC8 | Q9BY41 | 6/20 | 0.33 |
| ▸ | HDAC6 | Q9UBN7 | 6/20 | 0.33 |
| ▸ | HDAC9 | Q9UKV0 | 6/20 | 0.33 |
| ▸ | HDAC5 | Q9UQL6 | 6/20 | 0.33 |
| ▸ | HDAC10 | Q969S8 | 5/20 | 0.33 |
| ▸ | NCOR2 | Q9Y618 | 2/20 | 0.33 |
| ▸ | HPGD | P15428 | 1/20 | 0.33 |
| ▸ | SMN1; SMN2 | Q16637 | 1/20 | 0.33 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL5412235 | 0.77 | GAA (0.37) | MAPTKDM4EGAARAB9ASMN1; SMN2 | |
| SCHEMBL3289607 | 0.72 | POLB (0.48) | MAPTRAB9ASMN1; SMN2 | |
| SCHEMBL4481007 | 0.70 | MAPT (0.42) | MAPTKDM4EGAAMEN1KMT2A | |
| SCHEMBL9385508 | 0.69 | GAA (0.43) | MAPTGAA | |
| SCHEMBL27801775 | 0.69 | MAPT (0.43) | MAPTGAARAB9ASMN1; SMN2 | |
| SCHEMBL9381899 | 0.68 | SMN1; SMN2 (0.50) | MAPTKDM4EGAARAB9AMEN1 | |
| SCHEMBL5414764 | 0.66 | MAPT (0.41) | MAPTKDM4EGAARAB9AMEN1 | |
| SCHEMBL4915107 | 0.66 | GAA (0.37) | MAPTKDM4EGAARAB9AMEN1 | |
| SCHEMBL8900868 | 0.66 | GAA (0.38) | MAPTGAAHDAC1HDAC3HDAC4 | |
| SCHEMBL4788944 | 0.66 | KCNH3 (0.38) | MAPTKDM4EGAARAB9ASMN1; SMN2 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-2448961-A2 | TARGETS FOR RETROVIRUS ASSOCIATED DISEASES | Université de Liège (BE) | 2012-05-09 | — | — | EP | disclosed |
| US-20120090043-A1 | TARGETS FOR RETROVIRUS ASSOCIATED DISEASES | UNIVERSITE DE LIEGE (BE) | 2012-04-12 | — | — | US | disclosed |
| WO-2011000860-A2 | TARGETS FOR RETROVIRUS ASSOCIATED DISEASES | Université de Liège (BE) | 2011-01-06 | — | — | WO | disclosed |